SCHEMBL3687602

SCHEMBL3687602

COCCCn1c(=O)oc2ccc(-c3ccc(C[C@@H](C#N)NC(=O)[C@@H]4CCCCN4)cc3)cc21

nearest known ligand 0.72

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.72
CTSK P43235 3/20 0.59
KCNH2 Q12809 3/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3687606 1.00 CTSC (0.72) CTSCCTSKKCNH2
SCHEMBL2073466 0.96 CTSC (0.72) CTSCCTSKKCNH2
SCHEMBL2073462 0.96 CTSC (0.72) CTSCCTSKKCNH2
SCHEMBL7856284 0.89 CTSC (0.57) CTSCCTSKKCNH2
SCHEMBL2072323 0.87 CTSC (0.75) CTSCCTSKKCNH2
SCHEMBL2072320 0.87 CTSC (0.75) CTSCCTSKKCNH2
SCHEMBL290061 0.85 CTSC (0.73) CTSCKCNH2
SCHEMBL12422430 0.84 CTSC (0.57) CTSCCTSKKCNH2
SCHEMBL24973921 0.84 CTSC (0.65) CTSCCTSKKCNH2
SCHEMBL15084032 0.84 CTSC (1.00) CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010142985-A1 SUBSTITUTED N-[1-CYANO-2-(PHENYL)ETHYL]PIPERIDIN-2-YLCARBOXMIDE COMPOUNDS 761 ASTRAZENECA AB (SE) 2010-12-16 WO disclosed