SCHEMBL3688593

SCHEMBL3688593

COc1ccc(C(=O)C=Cc2ccc(NCCN(C)C)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F3 P13726 2/20 0.64
MAOB P27338 8/20 0.62
MAPT P10636 4/20 0.61
NPC1 O15118 1/20 0.61
LMNA P02545 1/20 0.61
MAOA P21397 3/20 0.59
XDH P47989 2/20 0.59
MEN1 O00255 2/20 0.59
ALDH1A1 P00352 2/20 0.59
KMT2A Q03164 2/20 0.59
P4HB P07237 1/20 0.59
CALM1 P0DP23 1/20 0.59
RAB9A P51151 1/20 0.59
BCHE P06276 3/20 0.58
CYP1B1 Q16678 3/20 0.57
CYP1A1 P04798 2/20 0.57
HSPD1 P10809 1/20 0.56
TNFRSF1A P19438 1/20 0.56
HSPE1 P61604 1/20 0.56
CYP3A4 P08684 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3688596 1.00 F3 (0.64) F3MAOBMAPTNPC1LMNA
SCHEMBL3693312 1.00 F3 (0.64) F3MAOBMAPTNPC1LMNA
SCHEMBL3693412 1.00 F3 (0.64) F3MAOBMAPTNPC1LMNA
SCHEMBL3683962 0.89 CYP1B1 (0.55) F3MAOBMAPTNPC1LMNA
SCHEMBL3693304 0.89 ABCG2 (0.65) F3MAOBMAPTNPC1LMNA
SCHEMBL3683960 0.89 ABCG2 (0.65) F3MAOBMAPTNPC1LMNA
SCHEMBL3692091 0.87 BCHE (0.60) MAOBMAPTNPC1LMNAMAOA
SCHEMBL3692089 0.87 BCHE (0.60) MAOBMAPTNPC1LMNAMAOA
SCHEMBL3695023 0.87 BCHE (0.60) MAOBMAPTNPC1LMNAMAOA
SCHEMBL3685113 0.86 BCHE (0.58) F3MAOBMAPTNPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP claimed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed