SCHEMBL3689543

SCHEMBL3689543

COc1ccc(C(=O)C=Cc2ccccc2NCCN(C)C)c(OC)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 5/20 0.60
MAPT P10636 7/20 0.58
PDE4A P27815 1/20 0.57
PDE4B Q07343 1/20 0.57
PDE4C Q08493 1/20 0.57
PDE4D Q08499 1/20 0.57
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
NPC1 O15118 3/20 0.56
RAB9A P51151 3/20 0.56
TNFRSF1A P19438 1/20 0.52
MAPK1 P28482 2/20 0.52
USP2 O75604 1/20 0.52
TLR9 Q9NR96 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
XDH P47989 1/20 0.49
CYP1A1 P04798 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3688287 1.00 ABCG2 (0.60) ABCG2MAPTPDE4APDE4BPDE4C
SCHEMBL3694918 0.95 ABCG2 (0.59) ABCG2MAPTPDE4APDE4BPDE4C
SCHEMBL3697030 0.95 ABCG2 (0.59) ABCG2MAPTPDE4APDE4BPDE4C
SCHEMBL3697931 0.92 MAPT (0.57) ABCG2MAPTPDE4APDE4BPDE4C
SCHEMBL3684123 0.92 MAPT (0.57) ABCG2MAPTPDE4APDE4BPDE4C
SCHEMBL3688290 0.88 MAPT (0.58) ABCG2MAPTPDE4APDE4BPDE4C
SCHEMBL3687942 0.87 MAPT (0.56) ABCG2MAPTPDE4APDE4BPDE4C
SCHEMBL3682374 0.87 MAPT (0.56) ABCG2MAPTPDE4APDE4BPDE4C
SCHEMBL3684125 0.86 PDE4A (0.57) ABCG2MAPTPDE4APDE4BPDE4C
SCHEMBL3694922 0.83 MAPT (0.57) ABCG2MAPTPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP claimed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed