SCHEMBL3693647

SCHEMBL3693647

CCC(C)(Sc1cccc(NC(=O)C(c2ccc(CN3N=C(c4ccccc4)OCC3=O)cc2)C(C)C)c1)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.35
ACKR3 P25106 1/20 0.35
SLC16A3 O15427 1/20 0.34
SLC16A1 P53985 1/20 0.34
MCTS1 Q9ULC4 1/20 0.34
ITGB3 P05106 8/20 0.33
ITGA2B P08514 8/20 0.33
PARP1 P09874 1/20 0.33
FFAR2 O15552 1/20 0.33
BACE1 P56817 1/20 0.33
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
TTK P33981 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1193761 0.92 PPARG (0.38) MAOBACKR3SLC16A3SLC16A1MCTS1
SCHEMBL13660625 0.90 MAOB (0.36) MAOBACKR3SLC16A3SLC16A1MCTS1
SCHEMBL3693646 0.89 MAOB (0.35) MAOBACKR3SLC16A3SLC16A1MCTS1
SCHEMBL3701718 0.88 PTGES (0.40) MAOBMAPTKMT2A
SCHEMBL1193997 0.86 MAOB (0.37) MAOBACKR3ITGB3ITGA2BPARP1
SCHEMBL1177676 0.86 MAOB (0.37) MAOBACKR3ITGB3ITGA2BPARP1
SCHEMBL12871721 0.86 MAOB (0.36) MAOBACKR3ITGB3ITGA2BPARP1
SCHEMBL1178122 0.85 ACKR3 (0.40) MAOBACKR3SLC16A3SLC16A1MCTS1
SCHEMBL3690996 0.85 ACKR3 (0.38) MAOBACKR3SLC16A3SLC16A1MCTS1
SCHEMBL1193806 0.82 PTGES (0.42) MAOBACKR3ITGB3ITGA2BPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed