SCHEMBL3694

SCHEMBL3694

O=C(Nc1ccc2c(=O)cc(-c3nn[nH]n3)oc2c1)c1ccc(OCCCCc2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RUVBL1 Q9Y265 1/20 1.00
CYSLTR2 Q9NS75 16/20 0.74
CYSLTR1 Q9Y271 16/20 0.74
NR1H4 Q96RI1 2/20 0.74
ABCC4 O15439 1/20 0.74
ABCB11 O95342 1/20 0.74
PGR P06401 1/20 0.74
HTR1A P08908 1/20 0.74
AR P10275 1/20 0.74
CHRM1 P11229 1/20 0.74
DRD1 P21728 1/20 0.74
PTGS1 P23219 1/20 0.74
SLC6A2 P23975 1/20 0.74
PDE4A P27815 1/20 0.74
ADORA1 P30542 1/20 0.74
ADRA1A P35348 1/20 0.74
OPRM1 P35372 1/20 0.74
DRD3 P35462 1/20 0.74
SLC6A3 Q01959 1/20 0.74
GPR17 Q13304 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15547055 0.87 RUVBL1 (0.76) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4
SCHEMBL18870151 0.86 RUVBL1 (0.75) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4
Pranlukast SCHEMBL18058592 0.85 CYSLTR2 (1.00) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4
Pranlukast SCHEMBL29349894 0.85 CYSLTR2 (1.00) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4
Pranlukast SCHEMBL29749274 0.84 CYSLTR2 (1.00) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4
SCHEMBL6956086 0.80 RUVBL1 (0.67) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4
SCHEMBL6962842 0.80 RUVBL1 (0.66) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4
SCHEMBL8115074 0.75 RUVBL1 (0.60) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4
SCHEMBL6950678 0.74 RUVBL1 (0.59) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4
SCHEMBL7897057 0.74 RUVBL1 (0.59) RUVBL1CYSLTR2CYSLTR1NR1H4ABCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12633 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436924-B1 None US claimed
EP-4676956-A2 ANTI-STEM CELL FACTOR (SCF) AND ANTI-THYMIC STROMAL LYMPHOPOIETIN (TSLP) ANTIBODIES AND BISPECIFIC CONSTRUCTS Celldex Therapeutics, Inc. (US) 2026-01-14 EP claimed
EP-4678659-A1 MONOCLONAL ANTIBODY PREPARATION TARGETING TSLP Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2026-01-14 EP claimed
US-20260000646-A1 Inhibition of Oral Microbe Biofilms THE UNIVERSITY OF TOLEDO (US) 2026-01-01 US claimed
WO-2025264860-A2 METHODS OF TREATING POST-COVID AIRWAY DISEASE YALE UNIVERSITY (US) 2025-12-26 WO claimed
WO-2025244529-A1 DOSING REGIMEN OF AN EGFR BINDING AND/OR COMPLEMENT ACTIVATING ANTIBODY MERUS N.V. (NL) 2025-11-27 WO claimed
EP-4615506-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES Sahin, Fikret (TR) 2025-09-17 EP claimed
WO-2025122933-A1 METHODS FOR THE DETECTION AND TREATMENT OF HEMATOLOGIC MALIGNANCY ASSOCIATED HYPERINFLAMMATION CHILDRENS HOPSITAL MEDICAL CENTER (US) 2025-06-12 WO claimed
WO-2025122021-A1 COMPOUNDS FOR USE IN THE TREATMENT OF HEART FAILURE WITH PRESERVED EJECTION FRACTION (HFPEF), THROUGH TARGETING OF S100A9 AND CORRESPONDING DIMER PARTNER AND RECEPTORS I3S - INSTITUTO DE INVESTIGAÇÃO E INOVAÇÃO EM SAÚDE, ASSOCIAÇÃO (PT) 2025-06-12 WO claimed
WO-2025110687-A1 PHARMACEUTICAL COMPOSITION COMPRISING BEPOTASTINE AND PRANLUKAST 대원제약주식회사 2025-05-30 WO claimed
WO-1999052553-A1 METHODS AND COMPOSITIONS USING CETIRIZINE IN COMBINATION WITH LEUKOTRIENE INHIBITORS FOR TREATING CONDITIONS RESPONSIVE TO LEUKOTRIENE INHIBITION SEPRACOR INC. (US) 1999-10-21 WO claimed
WO-1999052554-A1 METHODS AND COMPOSITIONS USING TERFENADINE METABOLITES IN COMBINATION WITH LEUKOTRIENE INHIBITORS SEPRACOR INC. (US) 1999-10-21 WO claimed
WO-1999052555-A1 METHODS AND COMPOSITIONS USING NORASTEMIZOLE IN COMBINATION WITH LEUKOTRIENE INHIBITORS SEPRACOR INC. (US) 1999-10-21 WO claimed
WO-1999044592-A1 ANTI-ASTHMA THERAPY ALZA CORPORATION (US) 1999-09-10 WO claimed
WO-1999032125-A1 COMPOSITION FOR TREATING RESPIRATORY AND SKIN DISEASES, COMPRISING AT LEAST ONE LEUKOTRIENE ANTAGONIST AND AT LEAST ONE ANTIHISTAMINE SCHERING CORPORATION (US) 1999-07-01 WO claimed
CN-1210465-A Methods of treatment and pharmaceutical compositions MERCK & CO INC (US) 1999-03-10 CN claimed
US-5876760-A Granules containing pranlukast, process for producing the granules, and method of improving adhesiveness of pranlukast ONO PHARMACEUTICAL CO., LTD. (JP) 1999-03-02 US claimed
WO-1998041193-A1 PREPARATION OF POWDER AGGLOMERATES SCHERING CORPORATION (US) 1998-09-24 WO claimed
EP-0834314-A1 GRANULES CONTAINING PRANLUKAST, PROCESS FOR PRODUCING THE GRANULES, AND METHOD OF LOWERING COHESIVENESS OF PRANLUKAST ONO PHARMACEUTICAL CO., LTD. (JP) 1998-04-08 EP claimed
WO-1997028797-A1 METHOD OF TREATMENT AND PHARMACEUTICAL COMPOSION MERCK & CO., INC. (US) 1997-08-14 WO claimed