SCHEMBL3694072

SCHEMBL3694072

Cc1cc(CNC(=O)C(c2ccc(CN3N=C(c4ccccc4)OCC3=O)cc2)C2CCCC2)ccc1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 1/20 0.37
PTGES O14684 3/20 0.37
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MCHR1 Q99705 1/20 0.35
SRC P12931 1/20 0.35
HTR1E P28566 1/20 0.34
S1PR3 Q99500 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3698450 0.91 BDKRB2 (0.35) BDKRB2PTGESTP53CYP1A2CYP3A4
SCHEMBL1079989 0.89 BDKRB2 (0.41) BDKRB2TP53CYP1A2CYP3A4CYP2D6
Bicarbonate SCHEMBL1079990 0.88 BDKRB2 (0.43) BDKRB2TP53CYP1A2CYP3A4CYP2D6
SCHEMBL1081746 0.86 BDKRB2 (0.40) BDKRB2CYP3A4
SCHEMBL1178266 0.86 BDKRB2 (0.41) BDKRB2PTGESTP53CYP1A2CYP3A4
SCHEMBL12872101 0.86 BDKRB2 (0.41) BDKRB2PTGESTP53CYP1A2CYP3A4
SCHEMBL12871694 0.85 BDKRB2 (0.40) BDKRB2PTGESTP53CYP1A2CYP3A4
SCHEMBL1178490 0.84 BDKRB2 (0.36) BDKRB2PTGESTP53CYP1A2CYP3A4
Bicarbonate SCHEMBL3704950 0.84 C3AR1 (0.41) BDKRB2PTGESTP53
SCHEMBL1178681 0.84 MAOB (0.41) BDKRB2PTGESMCHR1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed