SCHEMBL3694243

SCHEMBL3694243

CC(C)N(CCO)C(=O)c1cc([N+](=O)[O-])cc([N+](=O)[O-])c1N(CCBr)CCOS(C)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
HPGD P15428 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HKDC1 Q2TB90 1/20 0.35
HTT P42858 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3689649 0.95 KMT2A (0.46) KMT2AMEN1HPGDNPSR1HKDC1
SCHEMBL3691099 0.91 KMT2A (0.42) KMT2AMEN1HPGDNPSR1HKDC1
SCHEMBL3688111 0.91 KMT2A (0.45) KMT2AMEN1HPGDNPSR1HKDC1
SCHEMBL17191295 0.91 KMT2A (0.50) KMT2AMEN1HPGDNPSR1HKDC1
SCHEMBL3688122 0.88 KMT2A (0.42) KMT2AMEN1HPGDNPSR1HKDC1
SCHEMBL3690192 0.87 KMT2A (0.41) KMT2AMEN1HPGDNPSR1HKDC1
SCHEMBL3692467 0.86 KMT2A (0.43) KMT2AMEN1HPGDNPSR1HKDC1
SCHEMBL3691003 0.86 KMT2A (0.42) KMT2AMEN1HPGDNPSR1HKDC1
SCHEMBL12102448 0.85 KMT2A (0.43) KMT2AMEN1HPGDNPSR1HKDC1
SCHEMBL2962259 0.84 ALDH1A1 (0.43) KMT2AMEN1HPGDNPSR1HKDC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010044685-A1 NITROPHENYL MUSTARD ALCOHOLS, THEIR CORRESPONDING PHOSPHATES AND THEIR USE AS TARGETED CYTOTOXIC AGENTS AUCKLAND UNISERVICES LIMITED (NZ) 2010-04-22 WO claimed
WO-2010044685-A1 NITROPHENYL MUSTARD ALCOHOLS, THEIR CORRESPONDING PHOSPHATES AND THEIR USE AS TARGETED CYTOTOXIC AGENTS AUCKLAND UNISERVICES LIMITED (NZ) 2010-04-22 WO disclosed