SCHEMBL3695620

SCHEMBL3695620

NC(=O)[C@@H](CCCCl)c1ccccc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.41
ACP3 P15309 1/20 0.38
MAOB P27338 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
CACNA2D1 P54289 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNB1 Q02641 1/20 0.35
CACNA1C Q13936 1/20 0.35
PADI1 Q9ULC6 3/20 0.35
PADI3 Q9ULW8 3/20 0.35
PADI4 Q9UM07 3/20 0.35
PADI2 Q9Y2J8 2/20 0.35
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 2/20 0.34
TSHR P16473 2/20 0.34
CYP2C19 P33261 2/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1850628 1.00 CNR2 (0.41) CNR2ACP3MAOBSIRT2SIRT1
Hydrochloric Acid SCHEMBL3805598 0.99 CNR2 (0.40) CNR2ACP3MAOBSIRT2SIRT1
SCHEMBL12462316 0.87 CNR2 (0.42) CNR2ACP3MAOBSIRT2SIRT1
SCHEMBL719784 0.87 CNR2 (0.45) CNR2ACP3CACNA2D1CACNA1BCACNB1
SCHEMBL3696793 0.87 CNR2 (0.45) CNR2ACP3CACNA2D1CACNA1BCACNB1
SCHEMBL195361 0.87 CNR2 (0.42) CNR2ACP3MAOBCACNA2D1CACNA1B
Hydrochloric Acid SCHEMBL195363 0.86 CNR2 (0.44) CNR2ACP3CACNA2D1CACNA1BCACNB1
SCHEMBL6017225 0.86 CYP1A2 (0.43) CNR2ACP3CYP1A2CYP3A4CYP2C9
SCHEMBL13457707 0.83 CNR2 (0.39) CNR2ACP3CACNA2D1CACNA1BCACNB1
SCHEMBL194961 0.83 RAB9A (0.38) CNR2CYP1A2CYP2C19MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010098496-A1 PROCESS FOR PRODUCING TETRAHYDROTRIAZOLOPYRIDINE DERIVATIVE EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-09-02 WO claimed
WO-2010098496-A1 PROCESS FOR PRODUCING TETRAHYDROTRIAZOLOPYRIDINE DERIVATIVE EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-09-02 WO disclosed
WO-2010098496-A1 PROCESS FOR PRODUCING TETRAHYDROTRIAZOLOPYRIDINE DERIVATIVE EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-09-02 WO disclosed