SCHEMBL3697267

SCHEMBL3697267

CN(Cc1cc(Sc2ccc(Cl)nc2)n(-c2ccccc2F)n1)C(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.48
SLC6A4 P31645 8/20 0.48
HTR2A P28223 1/20 0.39
SCN9A Q15858 5/20 0.37
SLC16A3 O15427 5/20 0.34
SLC16A1 P53985 5/20 0.34
SCN10A Q9Y5Y9 2/20 0.34
SCN5A Q14524 1/20 0.33
CNR2 P34972 1/20 0.32
SPR P35270 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3703228 0.94 HTR2C (0.45) HTR2CSLC6A4HTR2ASCN9ASLC16A3
SCHEMBL3700534 0.94 HTR2C (0.45) HTR2CSLC6A4HTR2ASCN9ASLC16A3
SCHEMBL3692811 0.94 HTR2C (0.45) HTR2CSLC6A4HTR2ASCN9ASLC16A3
SCHEMBL3029602 0.92 HTR2C (0.49) HTR2CSLC6A4HTR2ASLC16A3SLC16A1
SCHEMBL3701837 0.91 HTR2C (0.43) HTR2CSLC6A4HTR2ACNR2
SCHEMBL3699694 0.91 HTR2C (0.45) HTR2CSLC6A4HTR2ACNR2
SCHEMBL3696768 0.90 HTR2C (0.45) HTR2CSLC6A4HTR2ASLC16A3SLC16A1
SCHEMBL3695013 0.90 HTR2C (0.43) HTR2CSLC6A4HTR2A
SCHEMBL3696458 0.90 HTR2C (0.43) HTR2CSLC6A4HTR2A
SCHEMBL3695135 0.90 HTR2C (0.44) HTR2CSLC6A4HTR2ASLC16A3SLC16A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed