SCHEMBL3699165

SCHEMBL3699165

COc1cccc2c(C(O)CN3CCOC(CNC(Cc4ccccc4)C4=COCO4)C3)ccnc12

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.38
DRD4 P21917 9/20 0.37
ABCB1 P08183 2/20 0.34
CNR1 P21554 1/20 0.33
EPHA2 P29317 1/20 0.32
KDR P35968 1/20 0.32
EPHB4 P54760 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5648717 0.86 KCNH2 (0.47) DRD4KCNH2
SCHEMBL5252749 0.83 KCNH2 (0.39) CNR2ABCB1KCNH2
SCHEMBL3691027 0.78 CYP2D6 (0.33) CNR2KCNH2
SCHEMBL3691984 0.78 DRD4 (0.40) DRD4
SCHEMBL5265635 0.76 DRD4 (0.36) DRD4EPHA2KDREPHB4KCNH2
SCHEMBL3695685 0.74 DRD4 (0.30) DRD4
SCHEMBL5318472 0.72 KCNH2 (0.37) KCNH2
SCHEMBL5254761 0.72 SLC2A1 (0.40) KCNH2
SCHEMBL3687758 0.71 CNR2 (0.33) CNR2
SCHEMBL5254666 0.69 KCNH2 (0.57) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed