SCHEMBL3687758

SCHEMBL3687758

COc1cccc2c(C(CO)N3C4CCC3CC(NC(Cc3ccccc3)C3=COCO3)C4)ccnc12

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
HTR1A P08908 2/20 0.31
ADRA1D P25100 2/20 0.31
ADRA1A P35348 2/20 0.31
ADRA1B P35368 2/20 0.31
F11 P03951 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3691027 0.87 CYP2D6 (0.33) CNR2CYP2D6CYP2C19HSP90AA1HSP90AB1
SCHEMBL5649376 0.85 KCNH2 (0.38) CYP2D6ADRA1A
SCHEMBL5252749 0.81 KCNH2 (0.39) CNR2
SCHEMBL3694994 0.73
SCHEMBL5651599 0.72 KCNH2 (0.46)
SCHEMBL3698321 0.72 HCRTR1 (0.35) CYP2C19HTR1AADRA1DADRA1AADRA1B
SCHEMBL3688489 0.71 HTR1A (0.33) HTR1AADRA1DADRA1AADRA1B
SCHEMBL3699165 0.71 CNR2 (0.38) CNR2
SCHEMBL5430924 0.69 KCNH2 (0.35)
SCHEMBL5254761 0.67 SLC2A1 (0.40) HTR1AADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2239260-A1 Novel compounds with antibacterial activity Morphochem Aktiengesellschaft Für Kombinatorische Chemie (DE) 2010-10-13 EP disclosed