SCHEMBL3699392

SCHEMBL3699392

[CH2]c1ccc(-c2cc3cc(Cc4ccccc4)ccc3o2)cc1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.58
FFAR1 O14842 4/20 0.52
S1PR3 Q99500 3/20 0.48
MAOB P27338 3/20 0.48
KCNH2 Q12809 1/20 0.43
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
MMP12 P39900 1/20 0.41
MMP13 P45452 1/20 0.41
CYP26A1 O43174 1/20 0.40
CYP26B1 Q9NR63 1/20 0.40
APP P05067 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3699394 0.86 MAOB (0.63) S1PR1FFAR1S1PR3MAOBKCNH2
SCHEMBL1602885 0.83 S1PR1 (0.58) S1PR1FFAR1S1PR3MAOBKCNH2
SCHEMBL6470762 0.82 MAOB (0.62) S1PR1FFAR1MAOBMMP12MMP13
SCHEMBL16152985 0.76 S1PR1 (0.51) S1PR1FFAR1S1PR3MAOBKCNH2
SCHEMBL1602753 0.76 S1PR1 (0.57) S1PR1FFAR1S1PR3MAOBKCNH2
SCHEMBL5401392 0.74 FFAR1 (0.67) S1PR1FFAR1MAOBESR1ESR2
SCHEMBL29214203 0.74 FFAR1 (0.62) S1PR1FFAR1MAOBESR1ESR2
SCHEMBL19553497 0.74 FFAR1 (0.62) S1PR1FFAR1MAOBESR1ESR2
SCHEMBL1603237 0.74 S1PR1 (1.00) S1PR1S1PR3KCNH2
SCHEMBL1601933 0.73 S1PR1 (0.48) S1PR1FFAR1S1PR3MAOBKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2010522162-A 2010-07-01 JP claimed
EP-2121648-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX Pharmaceuticals, Inc. (US) 2009-11-25 EP claimed
WO-2007109334-A2 SIP RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-09-27 WO claimed