SCHEMBL369946

SCHEMBL369946

O=C(Nc1ccc(Oc2ncnc3cc4c(cc23)OCCOCCOCCO4)c(F)c1)c1cccn(-c2ccc(F)cc2)c1=O

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MET P08581 18/20 0.67
AXL P30530 3/20 0.62
ABL1 P00519 1/20 0.62
TYRO3 Q06418 1/20 0.62
MERTK Q12866 1/20 0.62
MST1R Q04912 1/20 0.58
RIPK3 Q9Y572 3/20 0.58
RIPK1 Q13546 2/20 0.56
LCK P06239 1/20 0.56
KIT P10721 1/20 0.56
KDR P35968 1/20 0.56
FLT3 P36888 1/20 0.56
RIPK2 O43353 1/20 0.56
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18040372 0.90 MET (0.54) METAXLABL1TYRO3MERTK
SCHEMBL10133667 0.89 MET (0.67) METAXLTYRO3MERTKRIPK3
SCHEMBL23749464 0.83 MET (0.65) METAXLABL1TYRO3MERTK
SCHEMBL370073 0.82 MET (0.53) METAXLABL1TYRO3MERTK
SCHEMBL368546 0.81 MET (0.65) METAXLMST1RKITKDR
SCHEMBL370094 0.80 MET (0.67) METKDR
SCHEMBL23749515 0.80 KDR (0.64) METAXLABL1TYRO3MERTK
SCHEMBL23662776 0.80 AXL (0.67) METAXLTYRO3MERTKKIT
SCHEMBL24196720 0.79 MET (0.75) METAXLABL1TYRO3MERTK
SCHEMBL30381625 0.79 MET (0.75) METAXLABL1TYRO3MERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593462-B1 NOVEL FUSED HETEROCYCLIC DERIVATIVES USEFUL AS C-MET TYROSINE KINASE INHIBITORS BETTA PHARMACEUTICALS CO LTD (CN) 2016-09-07 EP disclosed
US-9242991-B2 Substituted fused heterocycles as c-Met tyrosine kinase inhibitors BETTA PHARMACEUTICALS CO., LTD (CN) 2016-01-26 US disclosed
US-20130123286-A1 Novel Fused Heterocyclic Derivatives Useful as c-Met Tyrosine Kinase Inhibitors BETTA PHARMACEUTICALS CO., LTD. (CN) 2013-05-16 US disclosed
WO-2012006960-A1 NOVEL FUSED HETEROCYCLIC DERIVATIVES USEFUL AS c-MET TYROSINE KINASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130123286-A1 Novel Fused Heterocyclic Derivatives Useful as c-Met Tyrosine Kinase Inhibitors MET, RET, ABL1 MET 1/4885AXL 408/4885ABL1 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.