Pyrazole

Pyrazole

SCHEMBL369975

c1cn[nH]c1.c1cnc2scnc2c1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 1/20 0.36
PDK1 Q15118 1/20 0.34
POLB P06746 1/20 0.33
RIPK1 Q13546 1/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29393471 0.84
SCHEMBL12820 0.84
Hydrochloric Acid SCHEMBL28163755 0.82 ALDH1A1 (0.46) ALDH1A1HSD17B10PDK1POLBRIPK1
Pyrrole SCHEMBL28787213 0.81 ALDH1A1 (0.39) ALDH1A1HSD17B10PDK1POLBRIPK1
SCHEMBL28733170 0.79 ALDH1A1 (0.35) ALDH1A1HSD17B10PDK1RIPK1
Benzo[D]Thiazole SCHEMBL360258 0.78 ALDH1A1 (0.66) ALDH1A1HSD17B10RIPK1NPC1RAB9A
SCHEMBL518747 0.74 ALDH1A1 (0.39) ALDH1A1HSD17B10PDK1POLBNPC1
Piperidine SCHEMBL3628735 0.73 ALDH1A1 (0.36) ALDH1A1HSD17B10PDK1RIPK1
Quinoline SCHEMBL2027950 0.72 ALDH1A1 (0.65) ALDH1A1HSD17B10POLBNPC1RAB9A
Quinoline SCHEMBL28561469 0.70 ALDH1A1 (0.63) ALDH1A1HSD17B10POLBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007510-A1 COMPOUNDS FOR BINDING AND IMAGING AMYLOID PLAQUES AND THEIR USE BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-19 WO disclosed
WO-2012007510-A1 COMPOUNDS FOR BINDING AND IMAGING AMYLOID PLAQUES AND THEIR USE BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-19 WO disclosed