SCHEMBL370102

SCHEMBL370102

CCCCC(=O)Oc1ccccc1I

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.65
KDM4E B2RXH2 1/20 0.65
MEN1 O00255 1/20 0.65
RECQL P46063 1/20 0.65
POLM Q9NP87 2/20 0.48
POLK Q9UBT6 2/20 0.48
POLL Q9UGP5 2/20 0.48
POLH Q9Y253 2/20 0.48
ALOX15 P16050 1/20 0.44
PPARG P37231 1/20 0.42
PTGS2 P35354 2/20 0.42
POLB P06746 1/20 0.41
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
FABP7 O15540 1/20 0.40
FABP3 P05413 1/20 0.40
FABP5 Q01469 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27546336 0.94 KMT2A (0.57) KMT2AKDM4EMEN1RECQLPOLM
SCHEMBL30942571 0.94 KMT2A (0.57) KMT2AKDM4EMEN1RECQLPOLM
SCHEMBL8207207 0.90 MEN1 (0.51) KMT2AKDM4EMEN1RECQLPOLM
SCHEMBL16756230 0.88 KDM4E (0.75) KMT2AKDM4EMEN1RECQLPOLM
SCHEMBL15558838 0.86 KMT2A (0.56) KMT2AKDM4EMEN1RECQLPOLM
SCHEMBL15547583 0.84 KDM4E (0.71) KMT2AKDM4EMEN1RECQLPOLM
SCHEMBL15547682 0.84 KDM4E (0.71) KMT2AKDM4EMEN1RECQLPOLM
SCHEMBL15548749 0.83 KDM4E (0.69) KMT2AKDM4EMEN1RECQLPOLM
SCHEMBL16239240 0.83 KDM4E (0.69) KMT2AKDM4EMEN1RECQLPOLM
SCHEMBL15548684 0.83 KDM4E (0.69) KMT2AKDM4EMEN1RECQLPOLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3668599-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS Inflazome Limited (IE) 2020-06-24 EP disclosed
WO-2019034690-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2019-02-21 WO disclosed
EP-2593427-A1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN Pfizer Limited (GB) 2013-05-22 EP disclosed
WO-2012007883-A1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LIMITED (GB) 2012-01-19 WO disclosed