SCHEMBL3701898

SCHEMBL3701898

CN(Cc1cc(Sc2cccnc2)n(-c2ccccc2Cl)n1)C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.49
SLC6A4 P31645 7/20 0.49
SLC16A3 O15427 10/20 0.39
SLC16A1 P53985 9/20 0.39
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
HTR2A P28223 1/20 0.33
CCNE2 O96020 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3702432 0.92 HTR2C (0.45) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3690712 0.90 HTR2C (0.45) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3697749 0.88 HTR2C (0.45) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3029602 0.88 HTR2C (0.49) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL4128944 0.87 SLC16A3 (0.38) HTR2CSLC6A4SLC16A3SLC16A1MEN1
SCHEMBL3692821 0.86 HTR2C (0.49) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3696583 0.84 HTR2C (0.51) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3700571 0.84 HTR2C (0.47) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3706675 0.84 HTR2C (0.39) HTR2CSLC6A4HTR2A
SCHEMBL3700851 0.82 HTR2C (0.39) HTR2CSLC6A4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed