SCHEMBL3700571

SCHEMBL3700571

COc1cc(Sc2cc(CN(C)C(=O)OC(C)(C)C)nn2-c2ccccc2Cl)ccn1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.47
SLC6A4 P31645 7/20 0.47
SLC16A3 O15427 9/20 0.39
SLC16A1 P53985 8/20 0.39
HTR2A P28223 1/20 0.34
BRAF P15056 1/20 0.33
CHRM1 P11229 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4132125 0.89 SLC16A3 (0.40) HTR2CSLC6A4SLC16A3SLC16A1ALDH1A1
SCHEMBL3694434 0.84 HTR2C (0.48) HTR2CSLC6A4SLC16A3SLC16A1
SCHEMBL3700575 0.84 SLC16A3 (0.40) HTR2CSLC6A4SLC16A3SLC16A1BRAF
SCHEMBL3692821 0.84 HTR2C (0.49) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3029602 0.84 HTR2C (0.49) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3701898 0.84 HTR2C (0.49) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3696583 0.84 HTR2C (0.51) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3690039 0.82 HTR2C (0.42) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3698137 0.82 HTR2C (0.49) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3706235 0.79 HTR2C (0.49) HTR2CSLC6A4SLC16A3SLC16A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed