SCHEMBL370290

SCHEMBL370290

BCCC(C)(C(=O)OC)c1ccc(N)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
ALDH1A1 P00352 3/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 3/20 0.34
SSTR4 P31391 1/20 0.33
EPHX2 P34913 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CFTR P13569 1/20 0.33
LMNA P02545 1/20 0.33
ABL1 P00519 1/20 0.33
RECQL P46063 2/20 0.33
HPGD P15428 2/20 0.33
ALOX15 P16050 2/20 0.33
TSHR P16473 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9612065 0.79 CNR1 (0.48) ALDH1A1CYP2C19POLBGAAEPHX2
SCHEMBL11307423 0.74 GAA (0.36) ALDH1A1CYP2C19POLBGAAEPHX2
SCHEMBL296610 0.74 SSTR4 (0.40) CYP2C19POLBSSTR4NPC1HPGD
SCHEMBL371221 0.70 SMN1; SMN2 (0.43) CYP2D6CYP2C19SSTR4NPC1RAB9A
SCHEMBL11152774 0.70 CYP3A4 (0.42) CYP2D6SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL3638360 0.69 TSHR (0.40) CYP2C19POLBSSTR4NPC1HPGD
SCHEMBL942098 0.68 CYP3A4 (0.40) ALDH1A1CYP2C19LMNARECQLHPGD
SCHEMBL4022599 0.68 TSHR (0.39) CYP2C19POLBSSTR4NPC1RAB9A
SCHEMBL3640874 0.68 TSHR (0.39) SLC6A3ALDH1A1CYP2C19POLBSSTR4
SCHEMBL730091 0.67 CNR1 (0.48) ALDH1A1GAAEPHX2NR1H4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200982-B1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2012-03-14 EP disclosed