SCHEMBL370292

SCHEMBL370292

CCCCN(C(C)=O)C1CCN(CCC(C)(C(=O)O)c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 4/20 0.61
TACR2 P21452 4/20 0.53
TACR1 P25103 3/20 0.53
UBE2M P61081 9/20 0.47
DCUN1D1 Q96GG9 9/20 0.47
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
PTBP1 P26599 1/20 0.39
KCNH2 Q12809 1/20 0.39
CACNA1I Q9P0X4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL297448 0.94 TACR3 (0.68) TACR3TACR2TACR1UBE2MDCUN1D1
SCHEMBL295922 0.91 TACR3 (0.58) TACR3TACR2TACR1UBE2MDCUN1D1
SCHEMBL295534 0.88 TACR3 (0.58) TACR3TACR2TACR1UBE2MDCUN1D1
SCHEMBL297464 0.84 TACR2 (0.58) TACR3TACR2TACR1UBE2MDCUN1D1
SCHEMBL295480 0.84 TACR2 (0.71) TACR3TACR2TACR1UBE2MDCUN1D1
SCHEMBL8042308 0.80 TACR2 (0.51) TACR3TACR2TACR1UBE2MDCUN1D1
SCHEMBL296656 0.80 TACR3 (0.77) TACR3TACR2TACR1UBE2MDCUN1D1
SCHEMBL297453 0.80 TACR3 (0.77) TACR3TACR2TACR1UBE2MDCUN1D1
SCHEMBL8052979 0.80 TACR3 (0.55) TACR3TACR2TACR1UBE2MDCUN1D1
SCHEMBL297889 0.79 TACR3 (0.50) TACR3TACR2TACR1KCNH2CACNA1I

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200982-B1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2012-03-14 EP disclosed