SCHEMBL8052979

SCHEMBL8052979

CSN(C1CC1)C1CCN(CCC(C)(C(=O)O)c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 5/20 0.55
TACR2 P21452 5/20 0.55
TACR1 P25103 4/20 0.55
KCNH2 Q12809 1/20 0.42
CACNA1I Q9P0X4 1/20 0.42
CCR5 P51681 2/20 0.39
OPRM1 P35372 3/20 0.39
OPRL1 P41146 2/20 0.39
SCN1A P35498 1/20 0.39
SCN2A Q99250 1/20 0.39
SCN3A Q9NY46 1/20 0.39
UBE2M P61081 2/20 0.38
DCUN1D1 Q96GG9 2/20 0.38
CHRM2 P08172 1/20 0.37
CHRM3 P20309 1/20 0.37
HTR7 P34969 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8032648 0.89 TACR3 (0.53) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL8042308 0.88 TACR2 (0.51) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL297464 0.87 TACR2 (0.58) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL297327 0.85 TACR2 (0.52) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL295480 0.84 TACR2 (0.71) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL295922 0.83 TACR3 (0.58) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL296518 0.83 TACR2 (0.54) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL296271 0.81 TACR2 (0.51) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL297448 0.81 TACR3 (0.68) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL370292 0.80 TACR3 (0.61) TACR3TACR2TACR1KCNH2CACNA1I

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009033995-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-03-19 WO disclosed