SCHEMBL3707346

SCHEMBL3707346

NC(=O)c1ccc(F)c(C(O)c2c[nH]c3ncc(-c4ccccc4)cc23)c1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 10/20 0.52
CAMKK2 Q96RR4 5/20 0.47
GSK3B P49841 2/20 0.47
CDC7 O00311 1/20 0.47
PLK4 O00444 1/20 0.47
CHEK1 O14757 1/20 0.47
AURKA O14965 1/20 0.47
MAPK13 O15264 1/20 0.47
PDPK1 O15530 1/20 0.47
DYRK3 O43781 1/20 0.47
ROCK2 O75116 1/20 0.47
RPS6KA5 O75582 1/20 0.47
PRKD3 O94806 1/20 0.47
PAK4 O96013 1/20 0.47
CHEK2 O96017 1/20 0.47
ABL1 P00519 1/20 0.47
EGFR P00533 1/20 0.47
NTRK1 P04629 1/20 0.47
INSR P06213 1/20 0.47
LCK P06239 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3505863 0.91 BRAF (0.44) AXLCAMKK2EGFRCDK2KDR
SCHEMBL3507088 0.91 DYRK1A (0.44) AXLGSK3BCDC7PLK4CHEK1
SCHEMBL3712316 0.87 AXL (0.51) AXLCAMKK2GSK3BCDC7PLK4
SCHEMBL3505306 0.87 CSF1R (0.41) AXLCAMKK2GSK3BCDC7PLK4
SCHEMBL3707351 0.86 GSK3B (0.54) AXLCAMKK2GSK3BCDC7PLK4
SCHEMBL2890696 0.85 BRAF (0.43) AXLCAMKK2GSK3BCDC7PLK4
SCHEMBL3505623 0.85 BRAF (0.44) AXLCAMKK2GSK3BPLK4AURKA
SCHEMBL3706478 0.83 CAMKK2 (0.37) AXLCAMKK2AURKARPS6KB1JAK3
SCHEMBL3504298 0.83 BRAF (0.35) AXLCAMKK2GSK3BPLK4AURKA
SCHEMBL2898883 0.82 CYP3A4 (0.44) AXLCAMKK2GSK3BCHEK1NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120122860-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122860-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS BRAF, RAF1, ARAF AXL 470/4885CAMKK2 497/4885GSK3B 3250/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.