SCHEMBL3707829

SCHEMBL3707829

Nc1nc(Cl)cc(C2CCN(C(=O)OCc3ccccc3)CC2)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.55
CYP2C19 P33261 1/20 0.55
TRPC3 Q13507 2/20 0.54
TRPC7 Q9HCX4 2/20 0.54
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
ENPP2 Q13822 3/20 0.48
GRIN2B Q13224 5/20 0.48
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47
DRD3 P35462 1/20 0.47
DHFR P00374 1/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7379278 0.89 SMN1; SMN2 (0.56) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL2881051 0.89 JAK2 (0.47) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
Guanidine SCHEMBL3709856 0.84 SMN1; SMN2 (0.54) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL16545218 0.83 SMN1; SMN2 (0.60) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL7411253 0.83 SMN1; SMN2 (0.60) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL3706053 0.80 HRH4 (0.53) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL13263856 0.80 TRPC3 (0.51) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL3708495 0.79 HRH4 (0.54) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL7374322 0.79 SMN1; SMN2 (0.57) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL12953174 0.78 TRPC3 (0.52) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010094721-A1 PIPERIDIN-PYRIMIDINE DERIVATIVES AS ANTAGONISTS OF HISTAMINE H4 RECEPTOR PALAU PHARMA, S. A. (ES) 2010-08-26 WO disclosed