SCHEMBL3708495

SCHEMBL3708495

Nc1nc(C2CCN(C(=O)OCc3ccccc3)CC2)cc(N2CCCNCC2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 4/20 0.54
HRH3 Q9Y5N1 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.46
CYP2C19 P33261 1/20 0.46
TRPC3 Q13507 2/20 0.46
TRPC7 Q9HCX4 2/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
SLC29A1 Q99808 1/20 0.45
GRIN2B Q13224 3/20 0.43
USP30 Q70CQ3 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
JAK2 O60674 2/20 0.41
JAK1 P23458 2/20 0.41
TYK2 P29597 2/20 0.41
JAK3 P52333 2/20 0.41
DHFR P00374 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3706053 0.81 HRH4 (0.53) HRH4SMN1; SMN2CYP2C19TRPC3TRPC7
SCHEMBL3707829 0.79 SMN1; SMN2 (0.55) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL606966 0.76 HRH4 (0.92) HRH4HRH3
Guanidine SCHEMBL3709856 0.76 SMN1; SMN2 (0.54) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
SCHEMBL605308 0.75 HRH4 (0.90) HRH4HRH3
SCHEMBL64989 0.74 MEN1 (0.59) SMN1; SMN2CYP2C19NPC1RAB9ASLC29A1
SCHEMBL16648631 0.73 SMN1; SMN2 (0.57) SMN1; SMN2CYP2C19TRPC3TRPC7NPC1
Hydrochloric Acid SCHEMBL28015140 0.73 MEN1 (0.58) SMN1; SMN2CYP2C19NPC1RAB9ASLC29A1
SCHEMBL3712220 0.73 HRH4 (0.55) HRH4HRH3
SCHEMBL603945 0.73 HRH4 (0.94) HRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010094721-A1 PIPERIDIN-PYRIMIDINE DERIVATIVES AS ANTAGONISTS OF HISTAMINE H4 RECEPTOR PALAU PHARMA, S. A. (ES) 2010-08-26 WO disclosed