SCHEMBL3708397

SCHEMBL3708397

Fc1ccc(-c2ncccc2CCl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.43
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
BCHE P06276 1/20 0.39
MAPK10 P53779 1/20 0.39
CACNA1B Q00975 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
PPARG P37231 1/20 0.36
NCOA2 Q15596 1/20 0.36
NCOA1 Q15788 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
TGFBR1 P36897 1/20 0.36
LIMK2 P53671 1/20 0.36
MAPK13 O15264 1/20 0.36
RAF1 P04049 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
DPP4 P27487 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719145 0.84 TRPV1 (0.47) MAPK14CYP1A2CYP2C19BCHEMAPK10
SCHEMBL4592340 0.84 KDM4E (0.41) CACNA1BPDE3BPDE3ALIMK2DPP4
SCHEMBL4600287 0.83 KCNA5 (0.43) LIMK2DPP4CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL9030551 0.82 TRPV1 (0.46) MAPK14CYP1A2CYP2C19BCHEMAPK10
SCHEMBL3711456 0.82 DPP4 (0.50) MAPK14CYP1A2CYP2C19BCHEMAPK10
SCHEMBL17456048 0.81 CYP11B1 (0.44) MAPK14LIMK2DPP4CYP11B1CYP11B2
SCHEMBL3907145 0.79 MAOB (0.44) MAPK14CYP1A2CYP2C19BCHEMAPK10
SCHEMBL11256542 0.79 BCHE (0.47) MAPK14BCHEMAPK10PDE3BPDE3A
SCHEMBL3906663 0.78 MAPK14 (0.40) MAPK14CYP1A2CYP2C19BCHEMAPK10
SCHEMBL8938109 0.78 MAPK14 (0.40) MAPK14CYP1A2CYP2C19BCHEMAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO claimed
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed