SCHEMBL3709845

SCHEMBL3709845

O=C1CNCCC1C(=O)OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
GLA P06280 1/20 0.43
HTR2C P28335 1/20 0.43
FABP7 O15540 1/20 0.43
FABP5 Q01469 1/20 0.43
FKBP1A P62942 1/20 0.42
ALDH1A1 P00352 2/20 0.41
NMT1 P30419 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27877768 0.99 TSHR (0.51) TSHRGLAHTR2CFABP7FABP5
SCHEMBL6631309 0.92 TSHR (0.47) TSHRGLAHTR2CFABP7FABP5
SCHEMBL988117 0.81 TSHR (0.51) TSHRFABP7FABP5FKBP1AALDH1A1
SCHEMBL1666324 0.78 CYP3A4 (0.52) TSHRFABP7FABP5FKBP1AALDH1A1
SCHEMBL606466 0.78 TSHR (0.55) TSHRHTR2CFABP7FABP5ALDH1A1
SCHEMBL19815901 0.78 HTR2C (0.46) TSHRGLAHTR2CFABP7FABP5
SCHEMBL2128136 0.77 MCL1 (0.56) TSHRFABP7FABP5FKBP1AALDH1A1
SCHEMBL5319406 0.77 MCL1 (0.56) TSHRFABP7FABP5FKBP1AALDH1A1
Hydrochloric Acid SCHEMBL3494457 0.77 TSHR (0.57) TSHRHTR2CFABP7FABP5ALDH1A1
SCHEMBL2300592 0.76 ALDH1A1 (0.46) TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391615-A1 Piperidine derivatives as nk3 receptor antagonists F. Hoffmann-La Roche AG (CH) 2011-12-07 EP disclosed
WO-2010086259-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-08-05 WO disclosed