SCHEMBL3710041

SCHEMBL3710041

O=C(NO)c1cc(NCc2ccccc2)nc(-c2ccc(C#Cc3cccnc3)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 9/20 0.46
HDAC6 Q9UBN7 5/20 0.46
HDAC3 O15379 4/20 0.46
HDAC2 Q92769 4/20 0.46
NCOR1 O75376 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 3/20 0.43
CLK4 Q9HAZ1 3/20 0.43
ALDH1A1 P00352 3/20 0.43
CYP2D6 P10635 2/20 0.43
HSD17B10 Q99714 2/20 0.43
FFAR1 O14842 1/20 0.43
ABCB1 P08183 1/20 0.42
ABCC1 P33527 1/20 0.42
ABCG2 Q9UNQ0 1/20 0.42
VCP P55072 1/20 0.42
USP2 O75604 1/20 0.41
CYP2C19 P33261 1/20 0.41
PTGES O14684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718158 0.89 HDAC1 (0.48) HDAC1HDAC6HDAC3HDAC2NCOR1
SCHEMBL3710406 0.88 PIK3CA (0.46) HDAC1CYP1A2CYP3A4CLK4ALDH1A1
SCHEMBL3716099 0.87 FFAR1 (0.41) HDAC1HDAC6HDAC3HDAC8ALDH1A1
SCHEMBL13188474 0.85 CAMK2D (0.47) HDAC1HDAC6HDAC3HDAC2FFAR1
SCHEMBL13188295 0.85 ABCB1 (0.48) HDAC1HDAC6HDAC3HDAC2NCOR1
SCHEMBL13188263 0.84 HDAC6 (0.42) HDAC1HDAC6HDAC3HDAC2NCOR1
SCHEMBL13187706 0.84 FGFR4 (0.39) HDAC1HDAC6HDAC3HDAC2NCOR1
SCHEMBL13188345 0.83 GRM5 (0.39) HDAC1HDAC6HDAC3HDAC2NCOR1
SCHEMBL3714241 0.83 HDAC6 (0.41) HDAC1HDAC6HDAC3HDAC2NCOR1
SCHEMBL3714333 0.82 HDAC1 (0.49) HDAC1HDAC6CYP1A2ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed