SCHEMBL3710139

SCHEMBL3710139

O=C(O)Nc1nc2ccc(-c3cncc(N4CCOCC4)c3)cc2s1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 10/20 0.56
PIK3CA P42336 3/20 0.56
PIK3CG P48736 7/20 0.54
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ABL1 P00519 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3711629 0.80 NPC1 (0.67) PIK3CAPIK3CGSMN1; SMN2
SCHEMBL13188391 0.78 PIK3CG (0.49) LRRK2PIK3CAPIK3CGABL1
SCHEMBL25258526 0.75 LRRK2 (0.58) LRRK2PIK3CAHTTSMN1; SMN2
SCHEMBL31114532 0.75 LRRK2 (0.58) LRRK2PIK3CAHTTSMN1; SMN2
SCHEMBL13188335 0.75 PIK3CG (0.69) LRRK2PIK3CAPIK3CGSMN1; SMN2
SCHEMBL3709559 0.75 PIK3CG (0.83) PIK3CAPIK3CGABL1
SCHEMBL3707938 0.75 PIK3CG (0.64) PIK3CAPIK3CGABL1
SCHEMBL3710994 0.75 PIK3CD (0.74) PIK3CAPIK3CGABL1
SCHEMBL13189097 0.74 PIK3CG (0.60) PIK3CAPIK3CGHTTSMN1; SMN2
SCHEMBL30697918 0.74 PIK3CA (0.70) LRRK2PIK3CAHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100144-A1 FUSED BICYCLIC COMPOUNDS AS INHIBITORS FOR PI3 KINASE MERCK SERONO S.A. (CH) 2010-09-10 WO disclosed