SCHEMBL3710259

SCHEMBL3710259

OCc1cnn(C2CC(n3cnc4c(N[C@H]5CCC[C@@H]5O)ncnc43)C(O)C2O)c1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 8/20 0.55
ADORA3 P0DMS8 6/20 0.55
ADORA2A P29274 5/20 0.55
CYP2D6 P10635 1/20 0.55
ADORA2B P29275 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3022704 1.00 ADORA1 (0.55) ADORA1ADORA3ADORA2ACYP2D6ADORA2B
SCHEMBL3027373 0.87 ADORA2A (0.57) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL3024769 0.86 ADORA2A (0.51) ADORA1ADORA3ADORA2ACYP2D6ADORA2B
SCHEMBL3129561 0.78 ADORA3 (0.50) ADORA1ADORA3ADORA2A
SCHEMBL3023215 0.78 ADORA3 (0.50) ADORA1ADORA3ADORA2A
SCHEMBL3022991 0.75 ADORA2A (0.58) ADORA1ADORA3ADORA2ACYP2D6ADORA2B
SCHEMBL3022156 0.73 ADORA2A (0.55) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL5399226 0.73 ADORA1 (0.72) ADORA1ADORA3ADORA2ACYP2D6ADORA2B
Gr-79236 SCHEMBL24436934 0.71 ADORA3 (1.00) ADORA1ADORA3ADORA2ACYP2D6ADORA2B
Gr-79236 SCHEMBL24437080 0.71 ADORA3 (1.00) ADORA1ADORA3ADORA2ACYP2D6ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205601-A1 PURINE DERIVATIVES AS ADENOSINE AL RECEPTOR LIGANDS Novartis Ag (CH) 2010-07-14 EP claimed
WO-2009050199-A1 PURINE DERIVATIVES AS ADENOSINE AL RECEPTOR LIGANDS NOVARTIS AG (CH) 2009-04-23 WO claimed