SCHEMBL3711569

SCHEMBL3711569

CC(=O)NCc1cncc(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.50
KDM4E B2RXH2 1/20 0.45
HDAC1 Q13547 2/20 0.44
HDAC6 Q9UBN7 1/20 0.44
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
PKM P14618 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP11B2 P19099 2/20 0.42
POLB P06746 2/20 0.42
HCAR2 Q8TDS4 1/20 0.42
SETDB1 Q15047 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3507481 0.84 SMN1; SMN2 (0.55) SMN1; SMN2KDM4EHDAC1MAPTHTT
SCHEMBL16213311 0.83 KDM4E (0.47) SMN1; SMN2KDM4EMAPTPKMPOLB
SCHEMBL14779720 0.83 SMN1; SMN2 (0.51) SMN1; SMN2KDM4EHDAC1MAPTHTT
SCHEMBL13632447 0.81 CYP2C9 (0.50) KDM4EHDAC1HDAC6MAPTKMT2A
SCHEMBL745029 0.80 SMN1; SMN2 (0.45) SMN1; SMN2KDM4EHDAC1MAPTHTT
SCHEMBL15926181 0.80 HDAC1 (0.50) KDM4EHDAC1HDAC6MAPTHTT
SCHEMBL22972298 0.79 NAMPT (0.49) HDAC1KMT2ACYP11B2HCAR2
SCHEMBL13999418 0.79 DYRK1A (0.49) SMN1; SMN2KDM4EHDAC1
SCHEMBL17695593 0.78 CYP11B2 (0.47) SMN1; SMN2KDM4EHDAC6MAPTKMT2A
SCHEMBL19323052 0.77 CYP11B2 (0.40) SMN1; SMN2KDM4EHDAC1HDAC6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100144-A1 FUSED BICYCLIC COMPOUNDS AS INHIBITORS FOR PI3 KINASE MERCK SERONO S.A. (CH) 2010-09-10 WO disclosed