SCHEMBL3711642

SCHEMBL3711642

CC(=O)Nc1cn2cc(-c3cncc(NS(C)(C)(=O)O)c3)ccc2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 11/20 0.53
PIK3CG P48736 3/20 0.52
PIK3CD O00329 2/20 0.52
PIK3CB P42338 2/20 0.52
PIK3C3 Q8NEB9 1/20 0.52
PI4KB Q9UBF8 1/20 0.52
BRAF P15056 5/20 0.46
MAPK13 O15264 4/20 0.46
KDR P35968 4/20 0.46
MAPK12 P53778 4/20 0.46
MAPK11 Q15759 4/20 0.46
MAPK14 Q16539 4/20 0.46
AKT1 P31749 1/20 0.46
MTOR P42345 1/20 0.46
MAP3K5 Q99683 1/20 0.43
PDGFRA P16234 2/20 0.43
IRAK4 Q9NWZ3 1/20 0.43
TGFBR1 P36897 1/20 0.43
ABL1 P00519 1/20 0.42
LRRK2 Q5S007 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8212993 0.82 PIK3CA (0.54) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3
SCHEMBL2946432 0.80 PIK3CA (0.65) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3
SCHEMBL3711646 0.79 PIK3CA (0.52) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3
SCHEMBL3252983 0.79 PIK3CA (0.55) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3
SCHEMBL3128211 0.78 PIK3CA (0.50) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3
SCHEMBL8214637 0.78 PIK3CA (0.60) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3
SCHEMBL13188706 0.78 PIK3CA (0.66) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3
SCHEMBL8216906 0.77 PIK3CA (0.71) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3
SCHEMBL13188708 0.75 PIK3C3 (0.61) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3
SCHEMBL14436388 0.73 PIK3CA (0.77) PIK3CAPIK3CGPIK3CDPIK3CBPIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100144-A1 FUSED BICYCLIC COMPOUNDS AS INHIBITORS FOR PI3 KINASE MERCK SERONO S.A. (CH) 2010-09-10 WO disclosed