SCHEMBL3712923

SCHEMBL3712923

COC(=O)Cc1cc2ccc(OC(F)(F)F)cc2[nH]c1=O

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 13/20 0.51
HSD17B10 Q99714 11/20 0.51
ALDH1A1 P00352 9/20 0.51
TSHR P16473 5/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
MAPT P10636 3/20 0.49
TP53 P04637 1/20 0.49
ALOX15 P16050 1/20 0.49
KMT2A Q03164 3/20 0.47
CYP1A2 P05177 1/20 0.47
MEN1 O00255 1/20 0.47
HPGD P15428 3/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718863 0.91 KDM4E (0.55) KDM4EHSD17B10ALDH1A1SMN1; SMN2MAPT
SCHEMBL3714878 0.86 KDM4E (0.46) KDM4EHSD17B10ALDH1A1TSHRSMN1; SMN2
SCHEMBL7073150 0.86 KDM4E (0.63) KDM4EHSD17B10ALDH1A1TSHRSMN1; SMN2
Trifluoroacetic Acid SCHEMBL7073292 0.81 KDM4E (0.45) KDM4EHSD17B10ALDH1A1TSHRSMN1; SMN2
SCHEMBL30548989 0.80 KDM4E (0.45) KDM4EHSD17B10ALDH1A1TSHRSMN1; SMN2
Trifluoroacetic Acid SCHEMBL7076651 0.80 KDM4E (0.46) KDM4EHSD17B10ALDH1A1TSHRSMN1; SMN2
SCHEMBL7071513 0.80 IDH1 (0.51) KDM4EHSD17B10ALDH1A1TSHRSMN1; SMN2
Trifluoroacetic Acid SCHEMBL7073477 0.79 CA12 (0.43) KDM4EHSD17B10ALDH1A1TSHRSMN1; SMN2
SCHEMBL3715876 0.79 EGFR (0.53) KDM4EHSD17B10ALDH1A1TSHRSMN1; SMN2
Trifluoroacetic Acid SCHEMBL7072029 0.77 HSD17B10 (0.46) KDM4EHSD17B10ALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393806-A1 INHIBITORS OF JUN N-TERMINAL KINASE Elan Pharmaceuticals Inc. (US) 2011-12-14 EP disclosed
WO-2010091310-A1 INHIBITORS OF JUN N-TERMINAL KINASE ELAN PHARMACEUTICALS, INC. (US) 2010-08-12 WO disclosed