SCHEMBL3713019

SCHEMBL3713019

COC(=O)c1cc(NC(=O)C2CCOCC2)nc(-c2ccc(C#Cc3ccc(CN4CCOCC4)nc3)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 7/20 0.42
DYRK1A Q13627 7/20 0.42
WNT1 P04628 5/20 0.40
JAK1 P23458 2/20 0.40
MOK Q9UQ07 4/20 0.38
ABL1 P00519 1/20 0.38
MAPK14 Q16539 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
HIF1A Q16665 1/20 0.37
EPAS1 Q99814 1/20 0.37
PIP5K1C O60331 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13188506 0.91 GSK3B (0.45) GSK3BDYRK1AWNT1JAK1MOK
SCHEMBL3714558 0.90 JAK1 (0.49) GSK3BDYRK1AJAK1
SCHEMBL3713032 0.85 MTOR (0.40) MOKMAPK14HIF1AEPAS1HRH3
SCHEMBL13188418 0.84 JAK1 (0.53) GSK3BDYRK1AJAK1ADORA3HIF1A
SCHEMBL3712780 0.83 ACP1 (0.49) MOKHIF1AEPAS1
SCHEMBL3713942 0.82 HRH3 (0.43) GSK3BDYRK1AWNT1MAPK14HIF1A
SCHEMBL3718978 0.81 HDAC1 (0.46) GSK3BDYRK1AWNT1ABL1MAPK14
SCHEMBL13188509 0.81 GSK3B (0.46) GSK3BDYRK1AWNT1JAK1ABL1
SCHEMBL3719071 0.80 MAPK1 (0.49) MOK
SCHEMBL3717690 0.78 HRH3 (0.44) GSK3BDYRK1AMAPK14HIF1AEPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed