SCHEMBL3713306

SCHEMBL3713306

O=CC[C@@]1(Cc2ccccc2)CCNC[C@H]1c1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 8/20 0.44
RCOR1 Q9UKL0 4/20 0.44
HTR3A P46098 1/20 0.34
MAOA P21397 6/20 0.33
MAOB P27338 6/20 0.33
KCNA5 P22460 1/20 0.32
SLC6A3 Q01959 2/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
REN P00797 2/20 0.32
CTSD P07339 1/20 0.32
CTSE P14091 1/20 0.32
PGC P20142 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3710752 1.00 KDM1A (0.44) KDM1ARCOR1HTR3AMAOAMAOB
SCHEMBL1439732 0.88 KDM1A (0.46) KDM1ARCOR1MAOAMAOBSLC6A3
SCHEMBL3708877 0.85 SLC6A2 (0.35) KDM1ARCOR1SLC6A3SLC6A2SLC6A4
SCHEMBL3715880 0.85 KDM1A (0.42) KDM1ARCOR1HTR3AMAOAMAOB
SCHEMBL3714347 0.82 KDM1A (0.48) KDM1ARCOR1HTR3AMAOAMAOB
SCHEMBL3712746 0.82 KDM1A (0.45) KDM1ARCOR1HTR3AMAOAMAOB
SCHEMBL3715321 0.82 KDM1A (0.45) KDM1ARCOR1HTR3AMAOAMAOB
SCHEMBL3644402 0.76 KDM1A (0.46) KDM1ARCOR1MAOAMAOB
SCHEMBL3712361 0.75 KDM1A (0.38) KDM1ARCOR1SLC6A4REN
SCHEMBL2225021 0.74 KDM1A (0.52) KDM1ARCOR1MAOAMAOBSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391615-A1 Piperidine derivatives as nk3 receptor antagonists F. Hoffmann-La Roche AG (CH) 2011-12-07 EP disclosed
WO-2010086259-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-08-05 WO disclosed