SCHEMBL3714347

SCHEMBL3714347

NCC[C@@]1(Cc2ccccc2)CCNC[C@@H]1c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 9/20 0.48
RCOR1 Q9UKL0 5/20 0.48
MAOA P21397 7/20 0.36
MAOB P27338 7/20 0.36
HTR3A P46098 1/20 0.35
SLC6A3 Q01959 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
REN P00797 2/20 0.32
CTSD P07339 1/20 0.32
CTSE P14091 1/20 0.32
PGC P20142 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3712746 0.88 KDM1A (0.45) KDM1ARCOR1MAOAMAOBHTR3A
SCHEMBL3715321 0.88 KDM1A (0.45) KDM1ARCOR1MAOAMAOBHTR3A
SCHEMBL3713306 0.82 KDM1A (0.44) KDM1ARCOR1MAOAMAOBHTR3A
SCHEMBL3710752 0.82 KDM1A (0.44) KDM1ARCOR1MAOAMAOBHTR3A
SCHEMBL1421527 0.80 KDM1A (0.52) KDM1ARCOR1MAOAMAOBSLC6A3
SCHEMBL2225021 0.80 KDM1A (0.52) KDM1ARCOR1MAOAMAOBSLC6A3
SCHEMBL3712361 0.80 KDM1A (0.38) KDM1ARCOR1SLC6A4REN
SCHEMBL3715880 0.80 KDM1A (0.42) KDM1ARCOR1MAOAMAOBHTR3A
SCHEMBL3710431 0.76 MEN1 (0.36) KDM1ARCOR1SLC6A3SLC6A2SLC6A4
SCHEMBL2017140 0.76 KDM1A (0.50) KDM1ARCOR1MAOAMAOBSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391615-A1 Piperidine derivatives as nk3 receptor antagonists F. Hoffmann-La Roche AG (CH) 2011-12-07 EP disclosed
WO-2010086259-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-08-05 WO disclosed