SCHEMBL3713327

SCHEMBL3713327

c1ccc(-c2n[nH]c(C3CNC3)n2)nc1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 2/20 0.58
TDP1 Q9NUW8 4/20 0.55
SMN1; SMN2 Q16637 4/20 0.55
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
L3MBTL1 Q9Y468 3/20 0.55
ALOX15 P16050 2/20 0.55
ALPL P05186 1/20 0.55
PKM P14618 1/20 0.55
HSD17B10 Q99714 1/20 0.55
KDM4E B2RXH2 5/20 0.46
AKT1 P31749 9/20 0.42
AKT2 P31751 9/20 0.42
HTT P42858 2/20 0.42
LMNA P02545 2/20 0.42
TP53 P04637 2/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3705458 0.98 USP30 (0.57) USP30TDP1SMN1; SMN2NPC1RAB9A
SCHEMBL10286741 0.85 USP30 (0.59) USP30TDP1SMN1; SMN2NPC1RAB9A
SCHEMBL3707946 0.78 AKT1 (0.44) USP30AKT1AKT2
SCHEMBL13256560 0.73 SMN1; SMN2 (0.55) TDP1SMN1; SMN2NPC1RAB9AL3MBTL1
SCHEMBL8311588 0.72 SMN1; SMN2 (1.00) TDP1SMN1; SMN2NPC1RAB9AL3MBTL1
Hydrochloric Acid SCHEMBL3706585 0.72 SMN1; SMN2 (0.54) TDP1SMN1; SMN2NPC1RAB9AL3MBTL1
SCHEMBL23488326 0.70 SMN1; SMN2 (0.66) USP30TDP1SMN1; SMN2NPC1RAB9A
SCHEMBL4562661 0.70 SMN1; SMN2 (0.66) USP30TDP1SMN1; SMN2NPC1RAB9A
SCHEMBL14446896 0.70 SMN1; SMN2 (0.66) TDP1SMN1; SMN2NPC1RAB9AL3MBTL1
SCHEMBL29210947 0.70 SMN1; SMN2 (0.66) USP30TDP1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396330-B1 FUSED PYRIMIDINES BAYER IP GMBH (DE) 2016-04-06 EP disclosed
EP-2396330-A1 FUSED PYRIMIDINES Bayer Pharma Aktiengesellschaft (DE) 2011-12-21 EP disclosed
WO-2010091808-A1 FUSED PYRIMIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-08-19 WO disclosed