SCHEMBL3714508

SCHEMBL3714508

CC(C)(C)OC(=O)N1C=C2CNCC2C1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
DDB1 Q16531 3/20 0.33
CRBN Q96SW2 3/20 0.33
NR1H2 P55055 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
ELANE P08246 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
ESR2 Q92731 1/20 0.32
RORC P51449 2/20 0.31
HSD11B1 P28845 1/20 0.31
NAMPT P43490 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18651951 0.82 KDM4E (0.38) KDM4EMAPTTHRBDDB1CRBN
SCHEMBL29728641 0.78 KDM4E (0.40) KDM4EMAPTTHRBDDB1CRBN
SCHEMBL29215624 0.74 GAA (0.37) KDM4EMAPTTHRBNR1H2CHRM2
SCHEMBL3806952 0.73 KDM4E (0.35) KDM4EMAPTTHRBDDB1CRBN
SCHEMBL2884871 0.71 KDM4E (0.39) KDM4EMAPTTHRBDDB1CRBN
SCHEMBL4876240 0.71 KDM4E (0.39) KDM4EMAPTTHRBDDB1CRBN
SCHEMBL3629917 0.71 KDM4E (0.39) KDM4EMAPTTHRBDDB1CRBN
SCHEMBL31339128 0.71 PARP1 (0.38) KDM4EMAPTTHRBDDB1CRBN
SCHEMBL7970964 0.68 CHRM2 (0.39) KDM4EMAPTTHRBDDB1CRBN
SCHEMBL2793465 0.67 USP2 (0.37) KDM4EMAPTTHRBDDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010108268-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2010-09-30 WO disclosed