SCHEMBL3715233

SCHEMBL3715233

O=C(O)C1N=c2ccccc2=CC1=O

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.31
TSHR P16473 1/20 0.31
NAPRT Q6XQN6 1/20 0.31
EP300 Q09472 1/20 0.31
KAT8 Q9H7Z6 1/20 0.31
ITGA4 P13612 1/20 0.30
ITGB7 P26010 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2778641 0.83 HTT (0.36) TSHRITGA4
SCHEMBL29056026 0.81 DAO (0.30) DAOTSHRNAPRT
SCHEMBL10726304 0.76 MEN1 (0.31)
SCHEMBL28201086 0.73
SCHEMBL28488959 0.72 MEN1 (0.30)
SCHEMBL27964340 0.72
SCHEMBL27669692 0.70 TSHR (0.33) DAOTSHRNAPRT
SCHEMBL28682085 0.69 GAA (0.34)
SCHEMBL7068822 0.68 DAO (0.34) DAOTSHRNAPRT
SCHEMBL30237619 0.68 PIM1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6897315-B2 Method for producing 8-methoxy-quinolinecarboxylic acids BAYER HEALTHCARE AKTIENGESELLSCHAFT (DE) 2005-05-24 US claimed
EP-1034173-B1 METHOD FOR PRODUCING 8-METHOXY-QUINOLINE CARBOXYLIC ACIDS BAYER HEALTHCARE AG (DE) 2005-04-27 EP claimed
US-20030208069-A1 Method for producing 8-methoxy-quinoline carboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 2003-11-06 US claimed
EP-0657448-B1 One pot process for the preparation of 3-quinolonecarboxylic acid derivatives BAYER AG (DE) 1998-03-04 EP claimed
US-5639886-A One-pot process for the preparation of 3-quinolonecarboxylic acid derivatives BAYER AKTIENGESELLSCHAFT (DE) 1997-06-17 US claimed
EP-0188194-B1 AMINOACRYLIC ACID DERIVATIVES BAYER AG (DE) 1990-07-04 EP claimed
CN-86100221-A AMINOACRYLIC ACID DERIVATIVES 1986-07-16 CN claimed
JP-2231476-A None JP disclosed
JP-7196621-A None JP disclosed
CN-113185505-B Quinolone oxazolidinone compound and preparation method and application thereof 中国农业大学 2022-09-27 CN disclosed
CN-114222839-A Antibacterial agent for high-pressure processing of fibers and high-pressure antibacterial processing method of fibers 大和化学工业株式会社 2022-03-22 CN disclosed
CN-113185505-A Quinolone oxazolidinone compound and preparation method and application thereof 中国农业大学 2021-07-30 CN disclosed
CN-111683930-A Novel isoxazole compound or salt thereof 日本欧爱特农业科技株式会社 2020-09-18 CN disclosed
CN-85101832-A The method for preparing 7-(3-aryl-1-piperazinyl)-3-quinolone carboxylic acid and 7-(3-encircles ethyl-1-piperazinyl)-3-quinolone carboxylic acid 1987-01-31 CN disclosed
CN-85101810-A 7-amido-1-cyclopropyl-6,8-dihalo-1,4-dihydro-4-oxo-3-quinoline carboxylic acid's preparation method 1987-01-17 CN disclosed
CN-86100221-A AMINOACRYLIC ACID DERIVATIVES 1986-07-16 CN disclosed
CN-86100221-A AMINOACRYLIC ACID DERIVATIVES 1986-07-16 CN disclosed
US-4404201-A N-/ /ALKANOYLAMINOALKANOYLAMINO OR AMINOALKANOYL AMINO/-DIHYDRO-OXO-3-QUINOLINYLCARBONYL/- DERIVATIVES WARNER-LAMBERT COMPANY (US) 1983-09-13 US disclosed
US-4382089-A Antibacterial amide compounds, compositions thereof and methods of using them WARNER-LAMBERT COMPANY (US) 1983-05-03 US disclosed
US-4374138-A PENICILLINS WARNER-LAMBERT COMPANY (US) 1983-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030208069-A1 Method for producing 8-methoxy-quinoline carboxylic acids QARS1, QPCT, PAM DAO 91/4885TSHR 4394/4885NAPRT 639/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.