SCHEMBL371585

SCHEMBL371585

COc1cc2nccc(Oc3ccc(NC(=N)CNC(=O)Cc4ccccc4)cc3F)c2cc1OC

nearest known ligand 0.74

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.74
KDR P35968 4/20 0.74
PDGFRB P09619 1/20 0.63
PDGFRA P16234 1/20 0.63
AXL P30530 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL411010 0.88 MET (0.81) METKDRPDGFRBPDGFRAAXL
SCHEMBL1882872 0.86 MET (0.84) METKDRPDGFRBPDGFRAAXL
SCHEMBL3457986 0.85 MET (1.00) METKDRPDGFRBPDGFRAAXL
SCHEMBL371908 0.83 MET (0.71) METKDR
SCHEMBL1879811 0.83 MET (0.78) METKDRPDGFRBPDGFRAAXL
SCHEMBL12444041 0.83 MET (0.73) METKDRPDGFRBPDGFRAAXL
SCHEMBL1484298 0.82 MET (0.69) METKDRPDGFRA
SCHEMBL5145179 0.82 MET (0.69) METKDRPDGFRBPDGFRAAXL
SCHEMBL371762 0.82 MET (0.69) METKDR
SCHEMBL1876439 0.82 MET (0.76) METKDRPDGFRBPDGFRAAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2409704-A2 c-Met modulators and methods of use Exelixis Inc. (US) 2012-01-25 EP disclosed