SCHEMBL3716168

SCHEMBL3716168

COc1nc(C2CC2)ccc1[N+](=O)[O-]

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TXNRD1 Q16881 10/20 0.45
MERTK Q12866 1/20 0.43
ALDH1A1 P00352 4/20 0.39
HTT P42858 2/20 0.39
TDP1 Q9NUW8 1/20 0.38
MAPT P10636 3/20 0.36
S1PR4 O95977 2/20 0.36
S1PR1 P21453 2/20 0.36
MAPK1 P28482 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
RAB9A P51151 1/20 0.36
GFER P55789 1/20 0.36
PAX8 Q06710 1/20 0.36
LMNA P02545 1/20 0.35
PIN1 Q13526 1/20 0.35
JAK2 O60674 1/20 0.35
HSP90AA1 P07900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31704071 0.79 TSHR (0.39) TXNRD1ALDH1A1TDP1MAPTMAPK1
SCHEMBL2132400 0.79 PRMT1 (0.42) ALDH1A1HTTMAPTMAPK1NPSR1
SCHEMBL2132394 0.79 PRMT1 (0.42) ALDH1A1HTTMAPTMAPK1NPSR1
SCHEMBL26868877 0.77 MERTK (0.48) TXNRD1MERTKALDH1A1HTTTDP1
SCHEMBL30666117 0.77 MERTK (0.48) TXNRD1MERTKALDH1A1HTTTDP1
SCHEMBL18188137 0.76 TXNRD1 (0.42) TXNRD1MERTKALDH1A1TDP1MAPT
SCHEMBL15471946 0.76 TDP1 (0.38) TXNRD1ALDH1A1TDP1MAPTMAPK1
SCHEMBL15514986 0.75 MERTK (0.49) TXNRD1MERTKALDH1A1HTTTDP1
SCHEMBL10740434 0.75 TXNRD1 (0.58) TXNRD1HTTMAPTS1PR4S1PR1
SCHEMBL29983153 0.75 MERTK (0.49) TXNRD1MERTKALDH1A1HTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010131146-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO disclosed
WO-2010131146-A1 CYCLOBUTENEDIONE DERIVATIVES PFIZER LIMITED (GB) 2010-11-18 WO disclosed