SCHEMBL3716448

SCHEMBL3716448

CN(C)c1ncc(-c2ccc(C#Cc3cccnc3)cc2)cc1C(=O)NO

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 2/20 0.42
MAP4K4 O95819 1/20 0.42
MINK1 Q8N4C8 1/20 0.42
FFAR1 O14842 1/20 0.40
PIK3C3 Q8NEB9 3/20 0.39
ADAM17 P78536 1/20 0.39
AAK1 Q2M2I8 2/20 0.39
GAK O14976 1/20 0.39
STK16 O75716 1/20 0.39
PIM1 P11309 1/20 0.39
AXL P30530 1/20 0.39
NEK2 P51955 1/20 0.39
STK3 Q13188 1/20 0.39
STK11 Q15831 1/20 0.39
BMP2K Q9NSY1 1/20 0.39
PTGES O14684 3/20 0.38
AKR1C3 P42330 2/20 0.38
SMPD1 P17405 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3709369 0.87 AAK1 (0.41) TNIKMAP4K4MINK1FFAR1PIK3C3
SCHEMBL13188601 0.87 SMPD1 (0.49) PIK3C3SMPD1HCRTR1HCRTR2HDAC1
SCHEMBL13188626 0.84 AAK1 (0.44) FFAR1PIK3C3ADAM17AAK1GAK
SCHEMBL3718656 0.84 CHRNA7 (0.41) TNIKFFAR1PIK3C3AAK1GAK
SCHEMBL3710648 0.81 SMPD1 (0.40) FFAR1ADAM17AAK1GAKSMPD1
SCHEMBL3716930 0.78 CCNE2 (0.43) GRM5
SCHEMBL3713525 0.78 MEN1 (0.43) FFAR1ADAM17AAK1SMPD1
SCHEMBL3711625 0.77 FFAR1 (0.36) TNIKFFAR1AAK1GAKSTK16
SCHEMBL3716655 0.76 FFAR1 (0.45) FFAR1SMPD1GRM5HDAC1HDAC6
SCHEMBL3713649 0.76 HDAC1 (0.52) TNIKFFAR1AAK1GAKSTK16

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed