SCHEMBL3716637

SCHEMBL3716637

O=C(O)C1CC(S(=O)(=O)c2ccccc2Cl)CN1C(=O)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSS P25774 15/20 0.67
CTSL P07711 8/20 0.67
CTSB P07858 4/20 0.67
RBP4 P02753 1/20 0.46
CTSK P43235 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3064915 1.00 CTSS (0.67) CTSSCTSLCTSBRBP4CTSK
SCHEMBL3061939 0.92 CTSS (0.58) CTSSCTSLCTSB
SCHEMBL696512 0.88 CTSS (0.64) CTSSCTSLCTSBCTSK
SCHEMBL696513 0.88 CTSS (0.64) CTSSCTSLCTSBCTSK
SCHEMBL3067551 0.87 CTSS (0.64) CTSSCTSLCTSBRBP4
SCHEMBL3065822 0.85 CTSS (0.53) CTSSCTSLCTSBCTSK
SCHEMBL3060759 0.84 CTSS (0.53) CTSSCTSLCTSBCTSK
SCHEMBL3067195 0.84 CTSS (0.52) CTSSCTSLCTSBCTSK
SCHEMBL3065895 0.83 CTSS (0.67) CTSSCTSLCTSB
SCHEMBL695458 0.82 CTSS (0.69) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed