SCHEMBL3717337

SCHEMBL3717337

CN(C)CCC(Nc1ncnc2c(C(=O)O)cccc12)c1cccc(NC(=O)c2ccc(F)cc2F)c1

nearest known ligand 0.87

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 19/20 0.87
AURKA O14965 19/20 0.87
AURKB Q96GD4 7/20 0.87

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL666814 0.93 RPS6KB1 (1.00) RPS6KB1AURKAAURKB
SCHEMBL3707136 0.90 RPS6KB1 (0.71) RPS6KB1AURKAAURKB
SCHEMBL16161983 0.89 AURKA (0.84) RPS6KB1AURKAAURKB
SCHEMBL666981 0.87 RPS6KB1 (1.00) RPS6KB1AURKAAURKB
SCHEMBL667258 0.86 AURKA (0.87) RPS6KB1AURKAAURKB
SCHEMBL3780777 0.86 AURKA (0.88) RPS6KB1AURKAAURKB
SCHEMBL666037 0.84 RPS6KB1 (0.85) RPS6KB1AURKAAURKB
SCHEMBL666799 0.84 RPS6KB1 (0.83) RPS6KB1AURKAAURKB
SCHEMBL666054 0.83 AURKA (0.86) RPS6KB1AURKAAURKB
SCHEMBL667095 0.83 RPS6KB1 (0.82) RPS6KB1AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396307-A1 NOVEL AMINO AZAHETEROCYCLIC CARBOXAMIDES Merck Patent GmbH (DE) 2011-12-21 EP claimed
WO-2010093419-A1 NOVEL AMINO AZAHETEROCYCLIC CARBOXAMIDES MERCK PATENT GMBH (DE) 2010-08-19 WO claimed