SCHEMBL3717850

SCHEMBL3717850

NC(=O)c1cccc(-c2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.74

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.74
PLG P00747 1/20 0.55
PLAU P00749 1/20 0.55
PLAT P00750 1/20 0.55
KIF11 P52732 5/20 0.54
ERN1 O75460 2/20 0.53
PDK2 Q15119 1/20 0.53
HDAC2 Q92769 1/20 0.52
P2RY14 Q15391 2/20 0.52
CCR6 P51684 1/20 0.52
AGXT P21549 1/20 0.49
PARP1 P09874 1/20 0.49
CCNE2 O96020 1/20 0.48
CCNE1 P24864 1/20 0.48
CDK2 P24941 1/20 0.48
SYK P43405 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3722990 0.98 DHODH (0.72) DHODHPLGPLAUPLATKIF11
SCHEMBL3727414 0.88 PLG (0.60) DHODHPLGPLAUPLATKIF11
SCHEMBL1348553 0.88 DHODH (0.60) DHODHPLGPLAUPLATKIF11
SCHEMBL30141887 0.87 DHODH (0.61) DHODHPLGPLAUPLATKIF11
SCHEMBL29917363 0.85 DHODH (0.71) DHODHKIF11PDK2HDAC2P2RY14
SCHEMBL177453 0.85 DHODH (0.71) DHODHKIF11PDK2HDAC2P2RY14
SCHEMBL3726477 0.84 DHODH (0.59) DHODHPLGPLAUPLATKIF11
SCHEMBL6999225 0.84 DHODH (0.63) DHODHERN1PARP1
SCHEMBL893254 0.83 DHODH (0.57) DHODHKIF11HDAC2SYK
SCHEMBL3018101 0.83 DHODH (0.57) DHODHPLGPLAUPLATKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US claimed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO claimed
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed