SCHEMBL3718137

SCHEMBL3718137

C[C@H]1C[N+](C(=O)[O-])(C(C)(C)C)CCN1C(=O)c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.42
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
TACR3 P29371 11/20 0.40
HSD11B1 P28845 2/20 0.38
TACR2 P21452 2/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719845 0.88 GAA (0.40) GHSRGAAHPGDCYP2C9CYP2C19
SCHEMBL3715353 0.88 GAA (0.40) GHSRGAAHPGDCYP2C9CYP2C19
SCHEMBL3714768 0.81 MEN1 (0.40) HSD11B1CA12CA1CA2CA7
SCHEMBL3713712 0.73 LIMK2 (0.42) HPGD
SCHEMBL4970907 0.72 DPP4 (0.31)
SCHEMBL2903872 0.70
SCHEMBL2904347 0.70
SCHEMBL3901950 0.70 GAA (0.51) GHSRGAAHPGDHSD11B1
SCHEMBL20370207 0.69 GAA (0.76) GAAHPGDHSD11B1CA12CA1
SCHEMBL16254905 0.68 GAA (0.84) GAAHPGDHSD11B1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010102663-A1 PIPERAZINE DERIVATIVES FOR USE IN THERAPY GLAXO GROUP LIMITED (GB) 2010-09-16 WO disclosed