SCHEMBL3715353

SCHEMBL3715353

C[C@@H]1C[N+](C(=O)[O-])(C(C)(C)C)CCN1C(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
ACHE P22303 1/20 0.40
HPGD P15428 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.38
HTT P42858 1/20 0.38
SMO Q99835 3/20 0.38
GHSR Q92847 1/20 0.38
RBP4 P02753 1/20 0.38
TSHR P16473 3/20 0.37
RECQL P46063 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 2/20 0.37
POLB P06746 1/20 0.37
ADRB2 P07550 1/20 0.37
MAPT P10636 1/20 0.37
MEN1 O00255 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719845 1.00 GAA (0.40) GAAACHEHPGDL3MBTL1HTT
SCHEMBL3718137 0.88 GHSR (0.42) GAAHPGDGHSRCYP3A4CYP2C9
SCHEMBL3714768 0.83 MEN1 (0.40) L3MBTL1HTTTSHRALDH1A1MAPT
SCHEMBL3713712 0.82 LIMK2 (0.42) HPGDRBP4TSHRSMN1; SMN2ALDH1A1
SCHEMBL4970907 0.74 DPP4 (0.31)
SCHEMBL2904347 0.72
SCHEMBL19454030 0.70 HPGD (0.64) GAAACHEHPGDL3MBTL1SMO
SCHEMBL252505 0.68 ACHE (0.55) GAAACHEHPGDL3MBTL1HTT
SCHEMBL12812547 0.68 HPGD (0.75) GAAACHEHPGDL3MBTL1HTT
SCHEMBL1429978 0.68 PSEN1 (0.50) ACHETSHRALDH1A1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010102663-A1 PIPERAZINE DERIVATIVES FOR USE IN THERAPY GLAXO GROUP LIMITED (GB) 2010-09-16 WO disclosed