SCHEMBL3718240

SCHEMBL3718240

c1ccc(CN2C3CCC2COC3)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.55
CHRM4 P08173 1/20 0.55
CHRM5 P08912 1/20 0.55
ALDH1A1 P00352 2/20 0.49
HRH3 Q9Y5N1 1/20 0.48
LTA4H P09960 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
CHRNB2 P17787 1/20 0.46
CHRNA7 P36544 1/20 0.46
CHRNA4 P43681 1/20 0.46
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
OPRM1 P35372 1/20 0.44
OPRK1 P41145 1/20 0.44
KCNH2 Q12809 1/20 0.44
DRD2 P14416 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL637410 0.93 CHRM2 (0.51) CHRM2CHRM4CHRM5ALDH1A1LTA4H
SCHEMBL636999 0.92 CHRM2 (0.58) CHRM2CHRM4CHRM5ALDH1A1HRH3
SCHEMBL20483452 0.86 CHRM2 (0.64) CHRM2CHRM4CHRM5ALDH1A1HRH3
SCHEMBL3082036 0.84 CHRM2 (0.47) CHRM2CHRM4CHRM5ALDH1A1HRH3
SCHEMBL3076478 0.84 CHRM2 (0.47) CHRM2CHRM4CHRM5ALDH1A1HRH3
SCHEMBL3083479 0.84 CHRM2 (0.47) CHRM2CHRM4CHRM5ALDH1A1HRH3
SCHEMBL3311708 0.84 CHRM2 (0.54) CHRM2CHRM4CHRM5ALDH1A1HRH3
SCHEMBL22533414 0.83 LTA4H (0.43) CHRM2CHRM4CHRM5ALDH1A1LTA4H
SCHEMBL21548123 0.83 CHRM2 (0.43) CHRM2CHRM4CHRM5ALDH1A1LTA4H
SCHEMBL14023655 0.83 CHRM2 (0.43) CHRM2CHRM4CHRM5ALDH1A1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120854-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-10-21 WO disclosed
WO-2010120854-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-10-21 WO disclosed
EP-0230274-A2 Derivatives of 7-(azabicycloalkyl)-quinoloncarboxylic acid and -naphthyridoncarboxylic acid BAYER AG (DE) 1987-07-29 EP disclosed