SCHEMBL3718876

SCHEMBL3718876

O=C(Nc1ccncc1)Nc1ccc(-c2cc3nccn3c(N3CCOCC3)n2)cc1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTOR P42345 16/20 0.57
PIK3CA P42336 7/20 0.57
PIK3CG P48736 3/20 0.57
RAF1 P04049 1/20 0.51
BRAF P15056 1/20 0.51
PIK3CD O00329 2/20 0.51
PIK3R1 P27986 1/20 0.48
CYP2C8 P10632 1/20 0.48
PIK3CB P42338 1/20 0.48
ATR Q13535 1/20 0.48
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3728227 0.90 MTOR (0.55) MTORPIK3CAPIK3CGRAF1BRAF
SCHEMBL3724095 0.88 GAA (0.51) MTORPIK3CAPIK3CGRAF1BRAF
SCHEMBL3797372 0.88 RAF1 (0.53) MTORPIK3CAPIK3CGRAF1BRAF
SCHEMBL3722456 0.78 ATR (0.56) MTORPIK3CARAF1BRAFPIK3CD
SCHEMBL3726551 0.77 MTOR (0.79) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL27940479 0.75 MTOR (0.73) MTORPIK3CAPIK3CGRAF1BRAF
SCHEMBL3724894 0.74 MTOR (0.77) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL32400 0.73 MTOR (1.00) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL3721523 0.72 PIK3CA (0.75) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL28603707 0.72 MTOR (0.54) MTORPIK3CAPIK3CGPIK3CDPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120994-A2 UREIDOARYL-AND CARBAMOYLARYL-MORPHOLINO- PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESIS WYETH LLC (US) 2010-10-21 WO disclosed