SCHEMBL3719259

SCHEMBL3719259

CC(C)c1n[nH]c2c(NCc3cccc(F)c3F)nc(NC3CCC(N)CC3)nc12

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 20/20 0.52
CCNA2 P20248 16/20 0.52
CCNT1 O60563 4/20 0.52
CDK9 P50750 4/20 0.52
CDK5 Q00535 3/20 0.52
CDK5R1 Q15078 2/20 0.52
CDK1 P06493 1/20 0.52
CDK4 P11802 1/20 0.52
CCNB1 P14635 1/20 0.52
CCND1 P24385 1/20 0.52
CDK6 Q00534 1/20 0.52
CCNE1 P24864 19/20 0.46
CCNE2 O96020 17/20 0.45
CCNT2 O60583 2/20 0.45
CCNA1 P78396 15/20 0.44
CDK7 P50613 1/20 0.41
CCNH P51946 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718031 0.92 CDK2 (0.51) CDK2CCNA2CCNT1CDK9CDK5
SCHEMBL3793236 0.87 CDK2 (0.57) CDK2CCNA2CCNT1CDK9CDK5
SCHEMBL3719256 0.85 CDK2 (0.73) CDK2CCNA2CCNT1CDK9CDK5
SCHEMBL3715540 0.85 CDK2 (0.57) CDK2CCNA2CCNT1CDK9CDK5
SCHEMBL3718025 0.85 CDK2 (0.59) CDK2CCNA2CCNT1CDK9CDK5
SCHEMBL2913765 0.85 CDK2 (0.71) CDK2CCNA2CCNT1CDK9CDK5
SCHEMBL3793439 0.84 CDK2 (0.54) CDK2CCNA2CCNT1CDK9CDK5
SCHEMBL3719473 0.83 CDK2 (0.65) CDK2CCNA2CCNT1CDK9CDK5
SCHEMBL3719282 0.83 CDK2 (0.64) CDK2CCNA2CCNT1CDK9CDK5
SCHEMBL3718045 0.82 CDK2 (0.59) CDK2CCNA2CCNT1CDK9CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010139288-A1 5,7-DISUBSTITUTED 3-ISOPROPYLPYRAZOLO[4,3-D]PYRIMIDINES FOR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS C3 BIO GMBH (DE) 2010-12-09 WO disclosed