SCHEMBL3719403

SCHEMBL3719403

CN(C)CCOc1ccc(NC(=O)Nc2ccc(-c3nc4c(c(N5C6CCC5COC6)n3)CN(C)CC4)cc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTOR P42345 19/20 0.69
PIK3CA P42336 16/20 0.69
PIK3CG P48736 2/20 0.64
CYP3A4 P08684 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721912 0.94 MTOR (0.72) MTORPIK3CAPIK3CG
SCHEMBL3724051 0.90 MTOR (0.71) MTORPIK3CAPIK3CGCYP3A4
SCHEMBL3718837 0.89 MTOR (0.72) MTORPIK3CAPIK3CGCYP3A4
SCHEMBL3725697 0.87 MTOR (0.67) MTORPIK3CAPIK3CGCYP3A4
SCHEMBL3727062 0.84 MTOR (0.55) MTORPIK3CAPIK3CGCYP3A4
SCHEMBL3721353 0.82 PIK3CA (0.70) MTORPIK3CAPIK3CG
SCHEMBL1431094 0.82 PIK3CA (1.00) MTORPIK3CAPIK3CG
SCHEMBL628588 0.81 MTOR (0.82) MTORPIK3CAPIK3CG
SCHEMBL3718595 0.78 PIK3CA (0.57) MTORPIK3CAPIK3CG
SCHEMBL56279 0.78 MTOR (0.74) MTORPIK3CAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120991-A1 5, 6, 7, 8-TETRAHYDROPYRIDO[4,3-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR, PI3, AND HSMG-1 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH LLC (US) 2010-10-21 WO claimed
WO-2010120991-A1 5, 6, 7, 8-TETRAHYDROPYRIDO[4,3-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR, PI3, AND HSMG-1 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH LLC (US) 2010-10-21 WO disclosed