SCHEMBL3720550

SCHEMBL3720550

CCNc1ccc2nc(Oc3ccc(Oc4ccccn4)c(C)c3)ccc2c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN7A Q01118 6/20 0.48
KCNH2 Q12809 6/20 0.48
SCN5A Q14524 1/20 0.44
SCN2A Q99250 1/20 0.44
SCN8A Q9UQD0 1/20 0.44
PDE10A Q9Y233 1/20 0.37
MAP4K4 O95819 1/20 0.36
SCN9A Q15858 2/20 0.36
P2RX3 P56373 3/20 0.36
DRD1 P21728 2/20 0.36
PTGS2 P35354 1/20 0.36
P2RX7 Q99572 1/20 0.35
NOTUM Q6P988 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722566 1.00 SCN7A (0.48) SCN7AKCNH2SCN5ASCN2ASCN8A
SCHEMBL3717667 0.85 MAPT (0.34) SCN7AKCNH2SCN5APDE10AMAP4K4
SCHEMBL3720645 0.83 MAPT (0.39) MAP4K4
SCHEMBL3719589 0.82 MAPT (0.34) SCN7AKCNH2SCN5ASCN2ASCN8A
SCHEMBL3720723 0.82 MAPT (0.44) MAP4K4
SCHEMBL3720739 0.81 MAPT (0.39) SCN5ASCN9AP2RX3
SCHEMBL3720742 0.81 MAPT (0.37) SCN7AKCNH2SCN9AP2RX3PDE4B
SCHEMBL3724195 0.81 MCHR1 (0.40) DRD1
SCHEMBL3720648 0.81 MAPT (0.36) SCN7AKCNH2P2RX3
SCHEMBL3717035 0.80 SCN7A (0.46) SCN7AKCNH2SCN5ASCN2ASCN8A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed